Pharmaceuticals/Chemicals
Aromasin (Exemestane)
Exemestane · Exe · Suicidal AI
Steroidal (suicidal) aromatase inhibitor; permanently inactivates aromatase enzyme.
Pharmacokinetic summary
- Model tier
- Advanced (t½ + Cmax + Tmax + F)
- Half-life
- 0.9 days
- Cmax
- 57.6 ng/mL
- Tmax
- 0.1 days
- Bioavailability
- 5%
- Typical dose
- 6.25–25 mg