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Pharmaceuticals/Chemicals

Nebivolol

Bystolic

β1-selective blocker with nitric-oxide-mediated vasodilation; BP management on-cycle.

Pharmacokinetic summary

Model tier
Advanced (t½ + Cmax + Tmax + F)
Half-life
0.7 days
Cmax
11.6 ng/mL
Tmax
0.1 days
Bioavailability
54%
Typical dose
2.5–20 mg